A Method for the Deprotection of Alkylpinacolyl Boronate Esters

作者:Sun Jing; Perfetti Michael T; Santos Webster L*
来源:Journal of Organic Chemistry, 2011, 76(9): 3571-3575.
DOI:10.1021/jo200250y

摘要

A two-step procedure for deprotection of alkylpinacolyl boronate esters via transesterification with diethanolamine followed by hydrolysis was successfully developed with the advantages of tolerance to various functional groups, short reaction time, and ease of product isolation.

  • 出版日期2011-5-6
  • 单位Virginia Tech; 美国弗吉尼亚理工大学(Virginia Tech)