Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains

作者:Crawford Terry D; Tsui Vickie; Flynn E Megan; Wang Shumei; Taylor Alexander M; Cote Alexandre; Audia James E; Beresini Maureen H; Burdick Daniel J; Cummings Richard; Dakin Les A; Duplessis Martin; Good Andrew C; Hewitt Michael C; Huang Hon Ren; Jayaram Hariharan; Kiefer James R; Jiang Ying; Murray Jeremy; Nasveschuk Christopher G; Pardo Eneida; Poy Florence; Romero F Anthony; Tang Yong; Wang Jian; Xu Zhaowu; Zawadzke Laura E; Zhu Xiaoyu
来源:Journal of Medicinal Chemistry, 2016, 59(11): 5391-5402.
DOI:10.1021/acs.jmedchem.6b00264