科研之友
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摘要
A short, four-step synthesis of Boc-protected (S)-dolaphenine is described, starting from protected phenylalanyl glycine. The key step is the cyclization of an endothiodipeptide to give a thiazolyl triflate, which can be subjected to a palladium-catalyzed reduction with formic acid.
- 出版日期2011-12
