Microwave-Assisted Amidation of Arylacetic Acids by Reaction with 2-Aryl-ethylamines

作者:Alajos Gruen; Matyas Milen; Tamas Foeldesi; Peter Abranyi Balogh; Laszlo Drahos; Gyoergy Keglevich*
来源:Synthetic Communications, 2013, 43(11): 1491-1498.
DOI:10.1080/00397911.2011.642925

摘要

Twenty-five amides were synthesized in almost quantitative yields by microwave-assisted condensation of arylacetic acids and 2-aryl-ethylamines under solventless conditions. The N-arylethyl-arylacetylamides are intermediates of the corresponding isoquinoline derivates. Supplemental materials are available for this article. Go to the publisher%26apos;s online edition of Synthetic Communications (R) to view the free supplemental file.

  • 出版日期2013-6-3