摘要
Several N-acyl-2-benzoylaziridines were prepared conveniently in good to high yields (71-93%) and used in the preparation of 5-benzoyloxazolines (76-91%) by a regio- and stereo-controlled reaction in the presence of NaI as an efficient catalyst under microwave irradiation in short reaction times (5-10 mins). The structure of the regioisomeric product was confirmed by X-ray analysis.
- 出版日期2008-12