Discovery of fruquintinib, a potent and highly selective small molecule inhibitor of VEGFR 1, 2, 3 tyrosine kinases for cancer therapy

作者:Sun Qiaoling; Zhou Jinghong; Zhang Zheng; Guo Mingchuan; Liang Junqing; Zhou Feng; Long Jingwen; Zhang Wei; Yin Fang; Cai Huaqing; Yang Haibin; Zhang Weihan; Gu Yi; Ni Liang; Sai Yang; Cui Yumin; Zhang Meifang; Hong Minhua; Sun Junen; Yang Zheng; Qing Weiguo; Su Weiguo; Ren Yongxin
来源:Cancer Biology and Therapy, 2014, 15(12): 1635-1645.
DOI:10.4161/15384047.2014.964087