A Simple Large-Scale Synthesis of Cbz-Protected Taurylsulfonyl Azide

作者：Brouwer Arwin J; Liskamp Rob M J^*

来源：Synlett, 2011, (15): 2228-2230.

DOI：10.1055/s-0030-1261201

• sulfonyl azide
• sulfonyl chloride
• large-scale synthesis
• chemoselectivity
• sulfo-click reaction

A simple and efficient method for the large-scale synthesis of Cbz-taurylsulfonyl azide is described. This sulfonyl azide is accessible from taurine using three or four synthetic steps.

• 出版日期2011-9