Direct Arylations of 2H-Indazoles On Water

作者:Ohnmacht Stephan A; Culshaw Andrew J; Greaney Michael F*
来源:Organic Letters, 2010, 12(2): 224-226.
DOI:10.1021/ol902537d

摘要

The efficient palladium-catalyzed synthesis of a range of substituted 2H-Indazoles via C-H arylation Is reported. Reactions are performed on water and provide a direct and mild route toward 2,3-diaryl indazoles of widespread biological significance.

  • 出版日期2010-1-15