Sonogashira coupling using PdEnCat (TM): a copper-, phosphine-, amine- and microwave-free alternative to the preparation of arylalkynes

作者：Barros Jose C; Yaunner Ricardo S; de Souza Andrea Luzia F; da Silva Joaquim F M^*; Antunes Octavio A C

来源：Applied Organometallic Chemistry, 2011, 25(11): 820-823.

DOI：10.1002/aoc.1845

• Sonogashira reaction
• C-C coupling
• PdEnCat
• mGluR5

Sonogashira coupling of iodo- and bromoarenes and acetylenes using PdEnCat (TM) 30 in a phosphine-, copper-, amine-, and microwave-free system was developed, which allows for the preparation of a modulator of glutamate receptor mGluR5.

• 出版日期2011-11