Application of Dimethylaminomethylene Ketone in Heterocycles Synthesis: Synthesis of 2-(Isoxazolo, Pyrazolo, and Pyrimido) Substituted Analogs of 1,4-Benzodiazepin-5-carboxamides Linked through an Oxyphenyl Bridge

作者：Kaur Navjeet^*; Tyagi Ruchi; Srivastava Manish; Kishore D

来源：Journal of Heterocyclic Chemistry, 2014, 51(S1): E50-E54.

DOI：10.1002/jhet.1841

Versatility of dimethylaminomethylene ketone derivative of 2-(4-acetyl)-phenoxyl-5-carboxamido-1,4-benzodiazepin-5-(4-methylpiperazinyl)-carboxamide (6) was explored to provide an easy one-pot access to its 2-(isoxazolo, pyrazolo, and pyrimido) substituted analogs 8, 9, 10, 11, 12, and 13, respectively.

• 出版日期2014-8