Discovery of potent aryl-substituted 3-[(3-methylpyridine-2-carbonyl) amino]-2,4-dimethyl-benzoic acid EP4 antagonists with improved pharmacokinetic profile

作者:Blanco Maria Jesus; Vetman Tatiana; Chandrasekhar Srinivasan; Fisher Matthew J; Harvey Anita; Chambers Mark; Lin Chaohua; Mudra Daniel; Oskins Jennifer; Wang Xu Shan; Yu Xiao Peng; Warshawsky Alan M
来源:Bioorganic & Medicinal Chemistry Letters, 2016, 26(3): 931-935.
DOI:10.1016/j.bmcl.2015.12.057