Highly regioselective palladium-catalyzed direct alkenylation of thiazolo[3,2-b]-1,2,4-triazoles via C-H activation

作者：Liu, Wenjie; Wang, Shaohua^*; Zhan, Haiying; Lin, Juan; He, Peiling; Jiang, Yi

来源：Tetrahedron Letters, 2014, 55(25): 3549-3552.

DOI：10.1016/j.tetlet.2014.04.095

• Dehydrogenative cross-coupling
• Thiazolo[3,2-b]-1,2,4-triazole
• Alkenylation
• Regioselectivity
• C-H activation

An efficient and regioselective palladium-catalyzed oxidative cross-coupling reaction between thiazolo[3,2-b]-1,2,4-triazoles and alkenes has been developed. This protocol provides easy access to a variety of functionalized thiazolo[3,2-b]-1,2,4-triazole derivatives.

• 出版日期2014-6-18
• 单位广东药科大学