An efficient alkynylation of 4-thiazolidinone with terminal alkyne under C-H functionalisation

作者:Shaikh Mohammed Umar M; Mudaliar Sulochana S; Chikhalia Kishor H*
来源:RSC Advances, 2016, 6(56): 50780-50785.
DOI:10.1039/c6ra05015h

摘要

A method of palladium catalysed efficient alkynylation through the cross coupling reaction of terminal alkynes with the slightly more acidic C-H bonds of 4-thiazolidinone has been developed. This method allows the direct introduction of an ethynyl group into the 4-thiazolidinone moiety.

  • 出版日期2016