A novel redox-sensitive protecting group for boronic acids, MPMP-diol

作者：Yan J; Jin S; Wang BH^*

来源：Tetrahedron Letters, 2005, 46(49): 8503-8505.

DOI：10.1016/j.tetlet.2005.10.010

• boronic acid
• protecting group
• DDQ

A new boronic acid protecting group, 1-(4-methoxyphenyl)-2-methylpropane-1,2-diol (MPMP-diol), has been developed. Both protection and deprotection can be accomplished under mild conditions with quantitative conversions. The deprotection can be carried out using 2.3-dichloro-5,6-dicyano-1,4-benzoquinone (DDQ).

• 出版日期2005-12-5