A microwave-assisted, propylphosphonic anhydride (T3P (R)) mediated one-pot Fischer indole synthesis

作者：Desroses Matthieu; Wieckowski Krzysztof; Stevens Marc; Odell Luke R^*

来源：Tetrahedron Letters, 2011, 52(34): 4417-4420.

DOI：10.1016/j.tetlet.2011.06.053

• Fischer indole
• Microwave
• Propylphosphonic anhydride
• Heterocycles

A rapid, mild, and high yielding protocol for the Fischer indolization of arylhydrazines with T3P (R) under microwave irradiation is described. Significant features of this method include short reaction times and preparative ease.

• 出版日期2011-8-24