A mild and efficient method for the synthesis of vinylogous carbamates from alkyl azides

作者：Reddy DS^*; Rajale TV; Shivakumar K; Iqbal J

来源：Tetrahedron Letters, 2005, 46(6): 979-982.

DOI：10.1016/j.tetlet.2004.12.047

• alkyl azide
• enaminone
• hydrogenation

A mild and efficient one-pot method for the synthesis of vinylogous carbamates is reported starting from alkyl azides under a hydrogen atmosphere using 10% Pd/C. The resulting products are useful intermediates for the synthesis of heterocyclic compounds, natural products, and in peptidomimetics.

• 出版日期2005-2-7