A Novel Three-Component One-Pot Reaction Involving beta-Naphthol, Aldehydes, and Urea Promoted by TMSCl/NaI

作者:Sabitha Gowravaram*; Arundhathi K; Sudhakar K; Sastry B S; Yadava J S
来源:Journal of Heterocyclic Chemistry, 2010, 47(2): 272-275.
DOI:10.1002/jhet.328

摘要

Amidoalkyl naphthol derivatives have been synthesized in good yields in a one-pot condensation of beta-naphthol, aromatic aldehydes and urea in presence of TMSCl/NaI at room temperature. Ring closure of amidoalkyl naphthol derivatives occurred at 140 degrees C to afford 1,2-dihydro-1-arylnaphtho[1,2-e] [1,3]oxazin-3-one derivatives.

  • 出版日期2010-3