A useful synthesis of the Phe-Arg phosphinic acid dipeptide isostere

作者：Kende AS^*; Dong HQ; Liu XW; Ebetino FH

来源：Tetrahedron Letters, 2002, 43(28): 4973-4976.

DOI：10.1016/S0040-4039(02)00957-7

• phosphinic acid dipeptide
• PheP-Arg isostere
• methylenemalonate ester
• phosphinate conjugate addition

A modular Method for construction of polypeptides containing the Phe-Arg phosphinic acid isostere is described.

• 出版日期2002-7-8