A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels-Alder Reaction Promoted by Silicon Tetrachloride

Massa Antonio<sup>*</sup>; de Sio Vincenzo; Villano Rosaria; Acocella M Rosaria; Palombi Laura; Sellitto Giusi; Peduto Antonella; Filosa Rosanna; De Capraris Paolo; Scettri Arrigo

doi:10.1055/s-0028-1087677

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A New Approach to Di- and Tetrasubstituted 2,3-Dihydropyridin-4(1H)-ones through Aza-Diels-Alder Reaction Promoted by Silicon Tetrachloride

作者：Massa Antonio^*; de Sio Vincenzo; Villano Rosaria; Acocella M Rosaria; Palombi Laura; Sellitto Giusi; Peduto Antonella; Filosa Rosanna; De Capraris Paolo; Scettri Arrigo

来源：Synthesis, 2009, 2009(4): 643-649.

DOI：10.1055/s-0028-1087677

摘要

Silicon tetrachloride promotes an aza-Diels Alder reaction with a range of imines and Danishefsky's diene or an alkylated derivative, giving the desired products in good to excellent yields.