Gold(I)-catalyzed formation of dihydroquinolines and indoles from N-aminophenyl propargyl malonates

作者：Gronnier Colombe; Odabachian Yann; Gagosz Fabien^*

来源：Chemical communications, 2011, 47(1): 218-220.

DOI：10.1039/c0cc00033g

The use of [XPhosAu(NCMe)]SbF(6) in nitromethane at 100 degrees C allows the rapid and efficient formation of variously substituted dihydroquinolines, which can be subsequently converted into indoles by a rare photochemical rearrangement.

• 出版日期2011