A general route to the synthesis of indoloazocines using allyl bromides prepared from Morita-Baylis-Hillman adducts

作者：Pandey Garima; Kant Ruchir; Batra Sanjay^*

来源：Tetrahedron Letters, 2015, 56(7): 930-933.

DOI：10.1016/j.tetlet.2014.12.124

• Nitrogen heterocycles
• Allylamine
• Allyl bromide
• Morita Baylis Hillman
• Friedel Craft's

A general approach to the synthesis of (E)-5-(substituted) benzylidene-2,3,4,5-tetrahydro-1H-azocino[5,4-b]indol-6(7H)-ones via intramolecular Friedel Craft's reaction of allylamines prepared from tryptamine and allyl bromides is reported.

• 出版日期2015-2-11