Aryne approach towards 2,3-difluoro-10-(1H-1,2,3-triazol-1-yl)pyrido[1,2-a]indoles

作者：Kopchuk Dmitry S^*; Nikonov Igor L; Zyryanov Grigory V; Nosova Emiliya V; Kovalev Igor S; Slepukhin Pavel A; Rusinov Vladimir L; Chupakhin Oleg N

来源：Mendeleev Communications, 2015, 25(1): 13-14.

DOI：10.1016/j.mencom.2015.01.003

Reaction between 3-(2-pyridyl)-1,2,4-triazines and in situ generated 4,5-difluorobenzyne in toluene affords 2,3-difluoro-10-(1H-1,2,3-triazol-1-yl)pyrido[1,2-a]indoles. The structure of one representative compound was confirmed by X-ray diffraction analysis.

• 出版日期2015-2