Microwave-Assisted Palladium-Catalyzed Heterogeneous Vinylation of 2(1H)-Pyridones

作者：Singh Brajendra K; Cavalluzzo Claudia; De Maeyer Marc; Debyser Zeger; Parmar Virinder S; Van der Eycken Erik^*

来源：European Journal of Organic Chemistry, 2009, 2009(27): 4589-4592.

DOI：10.1002/ejoc.200900677

• Microwave chemistry
• Heterogeneous catalysis
• Nitrogen heterocyles
• Natural products

A mild and efficient microwave-assisted vinylation of 2(1H)-pyridones has been developed using potassium vinyltrifluoroborate with palladium on carbon as the catalyst. Various vinylating agents, Pd sources and solvents have been screened.

• 出版日期2009-9