A one-pot construction of acridones by rhodium catalyzed reaction of N-phenyl-2-(1-sulfonyl-1H-1,2,3-triazol-4-yl)aniline

作者：Xu Hua Dong^*; Pan Ying Peng; Ren Xin Tao; Zhang Ping; Shen Mei Hua

来源：Tetrahedron Letters, 2015, 56(48): 6734-6737.

DOI：10.1016/j.tetlet.2015.10.059

• Acridone
• N-Sulfonyl 1,2,3-trizaole
• Rhodium carbene
• Cyclization
• Aza-vinyl metal carbene

A one-pot synthesis of N-alkyl acridone via rhodium catalyzed decomposition of N-phenyl-2-(1-sulfonyl-1H-1,2,3-triazol-4-yl)aniline and subsequent oxidative C-C bond fragmentation has been developed. 14 examples are presented and the yields range from 30% to 80%.

• 出版日期2015-12-2
• 单位常州大学