Asymmetric 1,3-dipolar cycloaddition reaction of azomethine imines to allyl alcohol

作者:Kato Tomomitsu; Fujinami Shuhei; Ukaji Yutaka*; Inomata Katsuhiko
来源:Chemistry Letters, 2008, 37(3): 342-343.
DOI:10.1246/cl.2008.342

摘要

The asymmetric 1,3-dipolar cycloaddition of azomethine imines to allyl alcohol was achieved by utilizing diisopropyl (R,R)-tartrate as a chiral auxiliary to afford the corresponding optically active trans-pyrazolidines with excellent regio-, diastereo-, and enantioselectivities.

  • 出版日期2008-3-5