A convenient synthesis of pyrazole-substituted heterocycles

作者:Shaaban Mohamed R; Eldebss Taha M A; Darweesh Ahmed F; Farag Ahmad M*
来源:Journal of Chemical Research, 2010, (1): 8-11.
DOI:10.3184/030823409X12608188070442

摘要

(E)-1-(5-Methyl-1-phenylpyrazol-4-yl)-3-(N,N-dimethylamino)-2-propen-1-one reacts with hydrazine, hydroxylamine, guanidine and aminopyrazole derivatives to afford the corresponding 3,4'-bipyrazole, pyrazolylisoxazole, pyrazolylpyrimidine and pyrazolo[1,5-a]pyrimidine derivatives, respectively. It reacts also with benzoquinone, naphthoquinone and N-benzoylglycine to give the corresponding benzofuran and pyrazolylpyranone derivatives, respectively.

  • 出版日期2010-1