A Remarkably Simple Protocol for the N-Formylation of Amino Acid Esters and Primary Amines

作者:Suchy Mojmir; Elmehriki Adam A H; Hudson Robert H E*
来源:Organic Letters, 2011, 13(15): 3952-3955.
DOI:10.1021/ol201475j

摘要

A simple, convenient, and wide scope protocol for the N-formylation of amino acid esters and primary amines has been developed utilizing only imidazole in warm DMF.

  • 出版日期2011-8-5