An Efficient Procedure for the Direct Nucleophilic Substitution of the Abiko-Masamune Auxiliary

作者：Li Jun; Li Pengfei; Menche Dirk^*

来源：Synlett, 2009, 2009(15): 2417-2420.

DOI：10.1055/s-0029-1217819

• synthetic methodology
• Lewis acid
• ester cleavage
• aldol reaction
• Abiko-Masamune auxiliary

An efficient method for the nucleophilic displacement of the Abiko-Masamune auxiliary is reported, which involves i-PrMgCl for intermediate ester activation.

• 出版日期2009-9-16