摘要

Asymmetric Friedel-Crafts reactions of indoles or pyrroles with coumarin-3-carboxylates catalyzed by Cu(OTf)(2) complexes with chiral bis(oxazoline) ligands have been developed. The highest ee (up to 82%) was achieved for indole with a nitro derivative of coumarin-3-carboxylate.

  • 出版日期2017-9