An Iron and Copper System Catalyzed C-H Arylation of Azoles with Arylboronic Acids

作者：Hu, Wei-Ye; Wang, Pei-Pei; Zhang, Song-Lin^*

来源：Synthesis (Germany), 2015, 47(1): 42-48.

DOI：10.1055/s-0034-1379073

• environmentally friendly
• copper and iron
• C-H activation
• azoles
• arylboronic acids

An efficient, environmentally friendly, and economical new method for arylation reactions of azoles with arylboronic acids via copper-iron-catalyzed C-H and C-B bond activation has been developed. The protocol tolerates a series of functional groups, such as methoxy, nitro, cyano, chloro, and trifluoromethyl groups.

• 出版日期2015-1
• 单位苏州大学