Advances in the Construction of 1-Monosubstituted 1,2,3-Triazole Ring

作者:Jiang Yubo*; Han Chunmei; Liang Xueqiu; Yang Peng; Wang Hong
来源:Chinese Journal of Organic Chemistry, 2013, 33(9): 1884-1890.
DOI:10.6023/cjoc201302025

摘要

As the 1,2,3-triazole derivatives were used in many expanding areas, its preparation has attracted much attention and obtained encouraging progress in recent years. The construction of the ring of monosubstituted 1,2,3-triazoles is more difficult than that of the other kinds of these heterocycles, owing to the special request for the structure of "alkyne source" and the relatively rigorous reaction conditions required in the system. This review covers the recent construction advances of the heterocycles based on the different moieties, such as acetylene, substituted acetylene, vinyl compounds, and others. Some important mechanisms were also discussed in details.

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