A new synthesis of substituted 2-trifluoromethylindoles

作者：Mokrushin Mikhail G; Shastin Aleksey V; Muzalevskiy Vasiliy M; Balenkova Elizabeth S; Nenajdenko Valentine G^*

来源：Mendeleev Communications, 2008, 18(6): 327-328.

DOI：10.1016/j.mencom.2008.11.014

The one-pot synthesis of substituted 2-trifluoromethylindoles from beta-halo-beta-(trifluoromethyl)-(o-halostyrene) and primary amines is based on a Cu(1)-catalysed double nucleophilic substitution reaction.

• 出版日期2008-12