A facile synthesis of 2-(N-alkylamino)-pyrimidin-4-one derivatives

作者:Li Jzhen*; Kou Jingping; Luo Xuyang; Fan Erkang
来源:Tetrahedron Letters, 2008, 49(17): 2761-2763.
DOI:10.1016/j.tetlet.2008.02.141

摘要

Substituted 2-(N-alkylamino)-pyrimidin-4-ones were synthesized using Pbf-activated thiourea. The six-membered pyrimidinones we TFA cleavage of the Pbf protecting group.