An efficient [3+2] cycloaddition for the synthesis of substituted pyrazolo[1,5-c]quinazolines

作者：Wang, Tao; Shao, Ailong; Feng, Haiyan; Yang, Shuwu; Gao, Meng^*; Tian, Jun; Lei, Aiwen

来源：Tetrahedron, 2015, 71(26-27): 4473-4477.

DOI：10.1016/j.tet.2015.03.019

• Pyrazolo[1,5-c]quinazolines
• Reagent-free
• Nitroolefins
• [3+2] Cycloaddition

A simple and efficient [3+2] cycloaddition reaction between N-iminoquinazolinium ylide and nitro-olefins was developed. From a synthetic point of view, this protocol represents an efficient way to pyrazolo[1,5-c]quinazolines derivatives.

• 出版日期2015-7-1
• 单位江西师范大学; 武汉大学