A novel and facile synthesis of 4-arylquinolin-2(1H)-ones under metal-free conditions

作者:Sun, Bin; Mai, Wen-Peng*; Yang, Liang-Ru; Mao, Pu; Yuan, Jin-Wei; Xiao, Yong-Mei
来源:Chinese Chemical Letters, 2015, 26(8): 977-979.
DOI:10.1016/j.cclet.2015.05.008

摘要

A novel and facile synthesis of 4-arylquinolin-2(1H)-ones without metal catalysis has been developed. This reaction involved cyclization/elimination steps and was performed under metal-free conditions using inexpensive reagents such as NaI, selectfluor and KOH.