New synthetic methodology leading to a series of novel heterocyclic alpha-aminophosphonates: a very attractive expansion of Kabachnik-Fields reaction

作者：Qu, Zhibo; Chen, Xiaolan^*; Yuan, Jinwei; Bai, Yunliang; Chen, Tong; Qu, Lingbo; Wang, Fujun; Li, Xu; Zhao, Yufen

来源：Tetrahedron, 2012, 68(15): 3156-3159.

DOI：10.1016/j.tet.2012.02.059

• One-pot
• Intramolecular cyclization
• Mechanism
• Heterocyclic alpha-Aminophosphonates
• Kabachnik-Fields reaction

A convenient one-pot three-component approach leading to synthesis of a series of novel heterocyclic alpha-aminophosphonates starting either from 2-hydroxyacetophenones or 2-hydroxybenzaldehyes was developed.

• 出版日期2012-4-15
• 单位河南工业大学; 厦门大学; 郑州大学