Discovery of spirocyclic proline tryptophan hydroxylase-1 inhibitors

作者:Goldberg Daniel R; De Lombaert Stephane; Aiello Robert; Bourassa Patricia; Barucci Nicole; Zhang Qing; Paralkar Vishwas; Valentine James; Zavadoski William
来源:Bioorganic & Medicinal Chemistry Letters, 2016, 26(4): 1124-1129.
DOI:10.1016/j.bmcl.2016.01.064