Direct arylation of benzoxazole C-H bonds with iodobenzene diacetates

作者:Yu Peng; Zhang Guangyou; Chen Fan*; Cheng Jiang
来源:Tetrahedron Letters, 2012, 53(34): 4588-4590.
DOI:10.1016/j.tetlet.2012.06.076

摘要

A Pd (OAc)(2)-catalyzed direct arylation of benzoxazole C-H bonds has been achieved with iodobenzene diacetates as the arylation reagent in moderate to good yields. The procedure tolerates a series of functional groups, such as methoxy, nitro, cyano, chloro, and bromo groups.