A borylative cyclisation towards indole boronic esters

作者:Huang Jianhui; Macdonald Simon J F; Harrity Joseph P A*
来源:Chemical communications, 2010, 46(46): 8770-8772.
DOI:10.1039/c0cc03577g

摘要

2-Alkynylaniline borylative cyclisations provide a direct means to access indole 3-boronic esters from simple precursors. The Pd-catalysed cyclisation can be merged with cross-coupling processes in the same reaction vessel, moreover, the products can be exploited in C-N bond forming reactions.

  • 出版日期2010