A convenient synthesis of chiral nonracemic vinyl aziridines

作者:Morton D; Pearson D; Field RA; Stockman RA*
来源:Organic Letters, 2004, 6(14): 2377-2380.
DOI:10.1021/ol049252l

摘要

The preparation of a range of alkyl and aryl chiral vinyl aziridines was achieved in high yield and stereoselectivity, and with excellent diastereoselectivity, by reaction of tert-butylsulfinylimines with the ylide derived from S-allyl tetrahydrothiophenium bromide.

  • 出版日期2004-7-8