Amino acid-mediated Goldberg reactions between amides and aryl iodides

作者：Deng W; Wang YF; Zou W; Liu L^*; Guo QX

来源：Tetrahedron Letters, 2004, 45(11): 2311-2315.

DOI：10.1016/j.tetlet.2004.01.119

• copper
• Goldberg reaction
• amide
• aryl halide
• coupling

A highly general, experimentally simple, and inexpensive catalyst system was developed for the amidation of aryl iodides by using 5 mol% of CuI as catalyst, 20 mol% of an amino acid as ligand, and K3PO4 as base.

• 出版日期2004-3-8
• 单位中国科学技术大学