Phenanthridine or isoquinoline are good reagents for the synthesis of enamino esters

作者:Nassiri Mahmoud; Heydari Reza; Hazeri Nourollah; Habibi Khorassani Sayyed Mostafa; Maghsoodlou Malek Taher*; Milani Forough Jalili
来源:Journal of Chemical Research, 2010, (7): 365-369.
DOI:10.3184/030823410X12767058123665

摘要

A new class of enamino esters has been isolated in excellent yields from the 1:1:1 addition reaction between phenanthridine or isoquinoline and activated acetylenic esters in the presence of heterocyclic NH compounds (succinimide, 5-nitroindazole, benzoxazolinone, 6-chlorobenzoxazolinone, carbazole and 3,6-dibromocabazole) or 1,3-dicarbonyl compounds such as 1,3-dimethylbarbituric acid and 1,3-diethy1-2-thiobar- bituric acid.

  • 出版日期2010-7