作者:Son Young Wook; Kwon Tae Hui; Lee Jae Kyun; Rae Ae Nim; Lee Jae Yeol; Cho Yong Seo*; Min Sun Joon
来源:Organic Letters, 2011, 13(24): 6500-6503.
DOI:10.1021/ol202792q
摘要
A concise synthesis of tetrabenazine and dihydrotetrabenazine is described. The key feature of this synthesis is the intramolecular aza-Prins-type cyclization of an amino allylsilane via oxidative C-H activation.