A Flexible Synthesis of Indoles from ortho-Substituted Anilines: A Direct Synthesis of Isocryptolepine

作者:Kraus George A*; Guo Haitao; Kumar Ganesh; Pollock Gerald III; Carruthers Heather; Chaudhary Divya; Beasley Jonathan
来源:Synthesis, 2010, (8): 1386-1393.
DOI:10.1055/s-0029-1218706

摘要

The reaction of anilines bearing a benzylic activating group in the ortho position with aromatic aldehydes or alpha,beta-unsaturated aldehydes results in an efficient synthetic route to substituted indoles.

  • 出版日期2010-4