A convenient Fischer indole synthesis of 2,3 '-biindoles

作者:Alford Philip E; Fu Liangfeng; Kubert Joseph K; Wang Lingshan; Gribble Gordon W*
来源:Tetrahedron Letters, 2011, 52(21): 2642-2644.
DOI:10.1016/j.tetlet.2011.03.049

摘要

Both symmetrical and unsymmetrical 2,3'-biindoles are efficiently synthesized in good to excellent yields by Fischer indole synthesis. The scope of the method was evaluated by examining substituent effects with para-substituted hydrazines and 3-acylindoles.

  • 出版日期2011-5-25