A Complementary Synthetic Approach to Fluorazone

作者:Calvert Matthew B; Sperry Jonathan*
来源:Journal of Heterocyclic Chemistry, 2014, 51(1): 282-284.
DOI:10.1002/jhet.2060

摘要

Pyrrole undergoes a regioselective zinc-mediated acylation with 2-bromobenzoyl chloride followed by a Cu-catalyzed N-arylation under microwave irradiation, delivering the important heteroaromatic of fluorazone.

  • 出版日期2014-1

全文