Discovery and Optimization of Selective Na(v)1.8 Modulator Series That Demonstrate Efficacy in Preclinical Models of Pain

作者:Bagal Sharan K; Bungay Peter J; Denton Stephen M; Gibson Karl R; Glossop Melanie S; Hay Tanya L; Kemp Mark I; Lane Charlotte A L; Lewis Mark L; Maw Graham N; Million William A; Payne C Elizabeth; Poinsard Cedric; Rawson David J; Stammen Blanda L; Stevens Edward B; Thompson Lisa R
来源:ACS Medicinal Chemistry Letters, 2015, 6(6): 650-654.
DOI:10.1021/acsmedchemlett.5b00059