An Efficient Synthesis of Aripiprazole, Buspirone and NAN-190 by the Reductive Alkylation of Amines Procedure

作者：Kowalski Piotr^*; Jaskowska Jolanta

来源：Archiv der Pharmazie, 2012, 345(1): 81-85.

DOI：10.1002/ardp.201100112

• Aripiprazole
• Buspirone
• NAN-190
• Reductive alkylation of amines
• Sodium triacetoxyborohydride

The reductive alkylation of amines procedure was applied for the synthesis of aripiprazole 1a, buspirone 1b, and NAN-190 1c.

• 出版日期2012-1