A concise synthesis of (-)-lentiginosine via an anti,syn-oxazine

作者：Kim Gun Woo; Jin Tian; Kim Jin Seok; Park Seok Hwi; Lee Kun Hee; Kim Seong Soo; Myeong In Soo; Ham Won Hun^*

来源：Tetrahedron: Asymmetry , 2014, 25(1): 87-91.

DOI：10.1016/j.tetasy.2013.11.009

A concise and stereocontrolled total synthesis of (-)-lentiginosine, a potent glycosidase inhibitor, has been achieved. Starting from anti,syn-oxazine as a chiral building block, the key features in these strategies are the Wittig reaction and cyclization.

• 出版日期2014-1-15